Dopaminergic Agents As Fibromyalgia Therapy

The treatment of fibromyalgia syndrome appears todopaminergic agent, pramipexole, with intriguing
be entering something of a golden age. Recently,results. Compared with the control group, patients in
after years of struggling just to be taken seriously,this study experienced gradual, significant
fibromyalgia patients have witnessed the release of aimprovement in measurements of pain, fatigue,
series of medications indicated for the treatment offunction, and overall well-being, suggesting that
fibromyalgia syndrome. While it is true that thesedopaminergic agents may be of value in the
medications are far from perfect and aren't effectivetreatment of fibromyalgia syndrome.(4)
for everyone, they have provided a strong sense ofWhile these results are encouraging, pramipexole is
direction for researchers and raised hopes for morenot yet approved for the treatment of fibromyalgia
efficacious treatments in the future.syndrome, and in the absence of an approved
Currently, the most promising areas of researchprescription product, some fibromyalgia patients have
center around central nervous systemturned to natural alternatives (dietary changes,
neurotransmittors and the role they play in painnatural supplements). Foods thought to affect
modulation. In the United States, the drugs currentlydopamine levels include almonds, bananas, avocados,
approved for the treatment of fibromyalgialima beans, pumpkin seeds and sesame seeds.
syndrome affect either the neurotransmitters,Unfortunately, despite anecdotal evidence reporting
serotonin and norepinephrine (duloxetine, milnacipran),positive results, no controlled studies exist to verify
or gamma-aminobutyric acid (pregabalin). These arethe efficacy of these efforts.
not the only neurotransmitters that are involved inThough research into the role of central nervous
pain modulation, however, leading researchers to looksystem neurotransmission in the expression of
at the role that dopamine may play in the pathologyfibromyalgia syndrome appears to hold great promise,
of fibromyalgia syndrome, too.the medications currently available are only marginally
In fact, there are several good reasons to think thateffective and the need for better therapies is acute.
dopamine may play a key role in the etiology andAs research progresses, dopaminergic agents such as
clinical presentation of fibromyalgia syndrome:pramipexole are likely to be added to the growing
1. A link has been identified between fibromyalgiaarsenal of approved agents, hopefully leading to
syndrome and an abnormality in a gene responsiblegreater relief for a growing number of fibromyalgia
for proper dopaminergic expression.(1) This geneticpatients.
link suggests that altered dopaminergic pathways1. Dan B, Hagit C, Lily N, Ebstein RP. An association
may be at least partially responsible for thebetween fibromyalgia and the dopamine D4 receptor
symptoms of fibromyalgia syndrome.exon III repeat polymorphism and relationship to
2. Studies utilizing positron emission topography (PET)novelty seeking personality traits. Molecular
to map brain response have empirically shown thatPsychiatry, 2004 9, 730-731.
fibromyalgia patients exhibit decreased dopaminergic2. Wood PB, Schweinhardt P, Jaeger E, Dagher A,
activity in response to painful stimuli when comparedHakyemez H, Rabiner E, Bushnell MC, Chizh BA.
to control groups.(2)(3) These fibromyalgia patientsFibromyalgia patients show an abnormal dopamine
also perceived the painful stimuli to be more severeresponse to pain. European Journal of Neuroscience,
than did the control group. Since dopamine has been2007 June;25(12):3576-3582.
implicated in both pain modulation and processing,3. Wood P, Patterson II J, Sunderland J, Tainter K,
these studies suggest dopamine may be at leastGlabus M, Lilien D. Reduced presynaptic dopamine
partially responsible for the widespread painactivity in fibromyalgia syndrome demonstrated with
experienced by fibromyalgia patients.positron emission tomography: a pilot study. The
3. Anecdotal evidence shows that low dopamineJournal of Pain, 8(1):51-58.
levels are associated with stiff, achy muscles,4. Holman AJ, Myers RR. A Randomized, Double-Blind,
cognitive impairment, and difficulty focusing. ThesePlacebo-Controlled Trial of Pramipexole, a Dopamine
symptoms are familiar to most fibromyalgia patients.Agonist, in Patients With Fibromyalgia Receiving
These are among the factors that have leadConcomitant Medications. Arthritis &
researchers to conduct clinical trials on theRheumatism, 2005 Aug;52(8):2495-2505.